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        產(chǎn)品名稱(chēng) A 1210477 from TOCRIS BIOSCIENCE
        產(chǎn)品貨號(hào) 6409/5
        產(chǎn)品價(jià)格 現(xiàn)貨詢(xún)價(jià),電話:010-67529703
        產(chǎn)品規(guī)格 5 mg
        產(chǎn)品品牌 TOCRIS BIOSCIENCE
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameA 1210477
        DescriptionSelective, high affinity Mcl-1 inhibitor (Ki = 454 pM). Disrupts Mcl-BIM complexes (IC50 in low μM range). Also inhibits Mcl-1NOXA interactions. Exhibits no effect on Bcl-XL-Bim or Bcl-X-BCL-Xs interactions. Induces apoptosis in multiple myeloma and non-small cell lung cancer cell lines and exhibits a synergistic effect with NavitoclaxTM to induce apoptosis in vitro. Cell permeable. Purity 98%. MW (observed): 850.04
        Size5 mg
        Concentrationn/a
        Applicationsn/a
        Other Names7-[5-[[4-[4-[(Dimethylamino)sulfonyl]-1-piperazinyl]phenoxy]methyl]-1,3-dimethyl-1H-pyrazol-4-yl]-1-[2-(4-morpholinyl)ethyl]-3-[3-(1-naphthalenyloxy)propyl]-1H-indole-2-carboxylic acid
        Gene, Accession, CAS #CAS: 1668553-26-1
        Catalog #6409/5
        Price
        Order / More InfoA 1210477 from TOCRIS BIOSCIENCE
        Product Specific Referencesn/a
        產(chǎn)品資料
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