| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | A 740003 |
| Description | Potent and selective P2X7 receptor antagonist (IC50 values are 18 and 40 nM for rat and human receptors respectively). Displays selectivity over a variety of P2X and P2Y receptors up to a concentration of 100 μM. Reduces nociception in animal models of persistent neuropathic and inflammatory pain. Also reduces neuroblastoma tumor growth in mice. Purity 98%. MW (observed): 474.55 |
| Size | 10 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | N-[1-[[(Cyanoamino)(5-quinolinylamino)methylene]amino]-2,2-dimethylpropyl]-3,4-dimethoxybenzeneacetamide |
| Gene, Accession, CAS # | CAS: 861393-28-4 |
| Catalog # | 3701/10 |
| Price | |
| Order / More Info | A 740003 from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 22185840, 22450808, 22898868, 23543737, 25682129, 26068648, 26542019, 27856358 |
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