| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | A 887826 |
| Description | Potent voltage-dependent NaV1.8 channel blocker (IC50 = 11 nM in recombinant human NaV1.8 channels). Reduces tactile allodynia in neuropathic rat models. 3- and 28-fold more potent at NaV1.8 channels compared to NaV1.2 and NaV1.7 channels respectively. Purity 97%. MW (observed): 480.99 |
| Size | 50 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 5-(4-Butoxy-3-chlorophenyl)-N-[[2-(4-morpholinyl)-3-pyridinyl]methyl-3-pyridine carboxamide |
| Gene, Accession, CAS # | CAS: 1266212-81-0 |
| Catalog # | 4249/50 |
| Price | |
| Order / More Info | A 887826 from TOCRIS BIOSCIENCE
|
| Product Specific References | PubMed: 24209626 |
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