| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | PF-573228 |
| Description | PF-573228 is a potent and selective inhibitor of focal adhesion kinase (FAK) (IC50 = 4 nM). PF-573,228 inhibits FAK phosphorylation on Tyr(397) with an IC50 of 30-100 nM. Displays 50 - 250-fold selectivity for FAK over other protein kinases. Blocks serum and fibronectin-directed migration and decreases focal adhesion turnover in vitro. MW: 491.49. Purity ≥98% by HPLC |
| Size | 10 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 3,4-Dihydro-6-[[4-[[[3-(methylsulfonyl)phenyl]methyl]amino]-5-(trifluoromethyl)-2-pyrimidinyl]amino]-2(1H)-quinolinone |
| Gene, Accession, CAS # | CAS: 869288-64-2 |
| Catalog # | 2819-10 |
| Price | |
| Order / More Info | PF-573228 from BIOVISION, INC. |
| Product Specific References | n/a |
| 產(chǎn)品資料 |
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