| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | NNC 05-2090 hydrochloride |
| Description | GABA uptake inhibitor that displays moderate selectivity for BGT-1 (mGAT-2) transporters (Ki values are 1.4, 15, 19 and 41 μM for hBGT-1, hGAT-3, hGAT-1 and hGAT-2 respectively). Anticonvulsive; inhibits sound-induced tonic and clonic convulsions in DBA/2 mice. Also displays affinity at α1- and D2-receptors (IC50 values are 266 and 1632 nM respectively). Purity 98%. MW (observed): 451.01 |
| Size | 10 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 1-[3-(9H-Carbazol-9-yl)propyl]-4-(2-methoxyphenyl)-4-piperidinol hydrochloride |
| Gene, Accession, CAS # | CAS: 184845-18-9 |
| Catalog # | 2747/10 |
| Price | |
| Order / More Info | NNC 05-2090 hydrochloride from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 26041994 |
| 產(chǎn)品資料 |
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