| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | AC 187 |
| Description | Orally active, potent amylin receptor antagonist (IC50 = 0.48 nM) that displays 38-fold and 400-fold selectivity over calcitonin and CGRP receptors respectively. Blocks amyloid β-induced neurotoxicity by attenuating the activation of initiator and effector caspases in vitro. Increases glucagon secretion, accelerates gastric emptying, alters plasma glucose levels and increases food intake in vivo. MW (observed): 2890.25. |
| Size | 500 ug |
| Concentration | n/a |
| Applications | n/a |
| Other Names | n/a |
| Gene, Accession, CAS # | CAS: 151804-77-2 |
| Catalog # | 3419/500U |
| Price | |
| Order / More Info | AC 187 from TOCRIS BIOSCIENCE
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| Product Specific References | PubMed: 24647952, 27688997 |
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