| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | AC 1903 |
| Description | Selective TRPC5 blocker (IC50 = 13.6 μM). Also displays weak inhibition at TRPC4 (IC50 >100 μM) but not TRPC6. Exhibits no effect against a standard panel of profiling kinases. Blocks TRPC5 channel activity in glomeruli of proteinuric rats. Suppresses severe proteinuria and prevents podocyte loss in a transgenic rat model of focal segmental glomerulosclerosis (FSGS). Purity 98%. MW (observed): 303.36 |
| Size | 25 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | N-(2-Furanylmethyl)-1-(phenylmethyl)-1H-benzimidazol-2-amine |
| Gene, Accession, CAS # | CAS: 831234-13-0 |
| Catalog # | 6766/25 |
| Price | |
| Order / More Info | AC 1903 from TOCRIS BIOSCIENCE
|
| Product Specific References | n/a |
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