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| Product Name | PFI-2 |
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| Description | PFI-2 is a novel potent and selective SETD7 histone lysine methyltransferase inhibitor (IC50 ~2 nM). It has > 100-fold selectivity over other methyltransferases and other non-epigenetic targets. PFI-2 has been shown to bind to SETD7 by ITC (Kd = 18 nM), and biotinylated PFI-2 interacts with SETD7 in pull-down studies. MW: 499.52. Purity ≥98% by HPLC |
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| Size | 5 mg |
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| Concentration | n/a |
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| Applications | n/a |
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| Other Names | (R)-8-fluoro-N-(1-oxo-1-(pyrrolidin-1-yl)-3-(3-(trifluoromethyl)phenyl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide |
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| Gene, Accession, CAS # | CAS: 1627676-59-8 |
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| Catalog # | B1259-5 |
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| Price | |
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| Order / More Info | PFI-2 from BIOVISION, INC. |
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| Product Specific References | n/a |
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