| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | DMP 543 |
| Description | Acetylcholine release stimulator. Potently enhances K+-stimulated [3H]-ACh release from rat hippocampal slices (EC50 = 700 nM), and increases release of dopamine and glutamate (EC50 values are 0.25 and 0.22 μM, respectively). Orally active in vivo; increases ACh levels in rats (with a minimum effective dose of 1 mg/kg) and exerts a long duration of action. More potent than linopirdine (Cat. No. 1999) both in vitro and in vivo. Also K+ channel blocker. Purity 99%. MW (observed): 412.44 |
| Size | 10 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 10,10-bis[(2-Fluoro-4-pyridinyl)methyl]-9(10H)-anthracenone |
| Gene, Accession, CAS # | CAS: 160588-45-4 |
| Catalog # | 2330/10 |
| Price | |
| Order / More Info | DMP 543 from TOCRIS BIOSCIENCE
|
| Product Specific References | PubMed: 21740972 |
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