| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | I-CBP112 |
| Description | I-CBP112 is a selective CBP/EP300 bromodomain inhibitor (IC50 values of 170 nM, 170 nM, 151 nM and 625 nM for CREBBP(Alphascreen), CREBBP(BLI), CREBBP(ITC) and EP300(ITC),respectively). Selective for CBP and p300 over ATAD2, BAZ2B, BRD2(2), BRD4(1), PB1(5), PCAF, PHIP(2) and TIF1α bromodomains in a BLI assay. MW: 468.59. Purity ≥98% by HPLC |
| Size | 1 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 1-[7-(3,4-Dimethoxyphenyl)-9-[[(3S)-1-methylpiperidin-3-yl]methoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one |
| Gene, Accession, CAS # | CAS: 1640282-31-0 |
| Catalog # | 9405-1 |
| Price | |
| Order / More Info | I-CBP112 from BIOVISION, INC. |
| Product Specific References | n/a |
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