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        產(chǎn)品名稱(chēng) IBMX from ARBOR ASSAYS, INC.
        產(chǎn)品貨號(hào) P019-1GM
        產(chǎn)品價(jià)格 現(xiàn)貨詢(xún)價(jià),電話(huà):010-67529703
        產(chǎn)品規(guī)格 1 gm
        產(chǎn)品品牌 ARBOR ASSAYS, INC.
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameIBMX
        DescriptionIBMX is a widely-used non-specific inhibitor of cyclic AMP and cyclic GMP phosphodiesterases (PDEs) with IC50s from 7 to 50 μM for PDE1-5, PDE7, and PDE11. PDE8A, PDE8B, and PDE9 are insensitive to IBMX. By inhibiting PDEs, IBMX increases cellular cAMP and cGMP levels, activating cyclic-nucleotide-regulated protein kinases. Methylxanthines, including IBMX, caffeine, and theophylline, bind adenosine receptors, typically antagonizing the suppressive effects of natural agonists. Suppresses alpha-adrenoceptor-mediated 5-HT release from neuroendocrine epithelial cells (IC50 = 1.3 μM).
        Size1 gm
        Concentrationn/a
        ApplicationsActivator or Inhibitor
        Other NamesPDE inhibitor
        Gene, Accession, CAS #n/a
        Catalog #P019-1GM
        Price
        Order / More InfoIBMX from ARBOR ASSAYS, INC.
        Product Specific Referencesn/a
        產(chǎn)品資料
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