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        產(chǎn)品名稱 FRAX597 from BIOVISION, INC.
        產(chǎn)品貨號 B1890-1
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格 1 mg
        產(chǎn)品品牌 BIOVISION, INC.
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameFRAX597
        DescriptionFRAX597 is a potent group I PAK (p21-activated kinase) inhibitor (IC50 values are 8, 13 and 19 nM for PAK1, 2 and 3, respectively). Displays significant inhibition of YES1, RET, CSF1R and TEK at 100 nM, but is inactive against group II PAK isoforms (IC50 >10 μM for PAK4). FRAX597 inhibits the proliferation of NF2-deficient schwannoma cells in culture and displays potent anti-tumor activity in vivo. MW: 558.1. Purity ≥98% by HPLC
        Size1 mg
        Concentrationn/a
        Applicationsn/a
        Other Names6-[2-Chloro-4-(5-thiazolyl)phenyl]-8-ethyl-2-[[4-(4-methyl-1-piperazinyl)phenyl]amino]pyrido[2,3-d]pyrimidin-7-(8H)-one
        Gene, Accession, CAS #CAS: 1286739-19-2
        Catalog #B1890-1
        Price
        Order / More InfoFRAX597 from BIOVISION, INC.
        Product Specific Referencesn/a
        產(chǎn)品資料
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