| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | SSR-240612 |
| Description | SSR-240612 is a potent and selective, non-peptide antagonist of the bradykinin B1 receptor (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors, respectively). It inhibits the contraction of rabbit aorta and rat ileum induced by the B1 receptor agonist des-Arg9-bradykinin (des-Arg9-BK) ex vivo in a concentration-dependent manner. MW: 793.4. Purity ≥98% by HPLC |
| Size | 5 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | (3R)-3-(1,3-benzodioxol-5-yl)-N-[(6-methoxy-2-naphthalenyl)sulfonyl]-β-alanyl-4-[[(2R,6S)-2,6-dimethyl-1-piperidinyl]methyl]-N-methyl-N-(1-methylethyl)-D-phenylalaninamide, monohydrochloride |
| Gene, Accession, CAS # | CAS: 464930-42-5 |
| Catalog # | B2349-5 |
| Price | |
| Order / More Info | SSR-240612 from BIOVISION, INC. |
| Product Specific References | n/a |
| 產(chǎn)品資料 |
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