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        產(chǎn)品名稱 PQ 69 from TOCRIS BIOSCIENCE
        產(chǎn)品貨號 5351/50
        產(chǎn)品價格 現(xiàn)貨詢價,電話:010-67529703
        產(chǎn)品規(guī)格 50 mg
        產(chǎn)品品牌 TOCRIS BIOSCIENCE
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NamePQ 69
        DescriptionPotent and selective A1 receptor inverse agonist. Exhibits high binding affinity at A1 receptor (Ki values are 0.07 and 0.96 nM for rat and human receptors respectively). Reduces basal [35S]-GTPγS binding 44.6% (IC50 = 0.19 nM). Antagonizes the effects of A1 agonist R-PIA (IC50 = 18.3 nM) and exhibits competitive antagonism on CCPA -induced tracheal contractions ex vivo. Displays 217- fold selectively over hA2A receptor and >1000-fold selectivity over hA3 receptor. Purity 98%. MW (observed): 350.39
        Size50 mg
        Concentrationn/a
        Applicationsn/a
        Other Names4-(Butylamino)-2-(3-fluorophenyl)-1,2-dihydro-3H-pyrazolo[4,3-c]quinolin-3-one
        Gene, Accession, CAS #CAS: 910045-32-8
        Catalog #5351/50
        Price
        Order / More InfoPQ 69 from TOCRIS BIOSCIENCE
        Product Specific Referencesn/a
        產(chǎn)品資料
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