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        產(chǎn)品名稱 MRK 016 from TOCRIS BIOSCIENCE
        產(chǎn)品貨號(hào) 3817/50
        產(chǎn)品價(jià)格 現(xiàn)貨詢價(jià),電話:010-67529703
        產(chǎn)品規(guī)格 50 mg
        產(chǎn)品品牌 TOCRIS BIOSCIENCE
        產(chǎn)品概述
        產(chǎn)品詳情
        Edit&nbsp
        Product NameMRK 016
        DescriptionGABAA receptor inverse agonist selective for the α5-subtype (EC50 = 3 nM). Exhibits affinity at benzodiazepine binding site of recombinant human GABAA receptors (Ki values are 0.77 nM, 0.83 nM, 0.85 nM and 1.4 nM for α3-, α1-, α2-, and α5-containing respectively). Increases long-term potentiation (LTP) in mouse hippocampal slices. Exhibits no anxiogenic or proconvulsant activity. Purity 98%. MW (observed): 368.39
        Size50 mg
        Concentrationn/a
        Applicationsn/a
        Other Names3-(1,1-Dimethylethyl)-7-(5-methyl-3-isoxazolyl)-2-[(1-methyl-1H-1,2,4-triazol-5-yl)methoxy]-pyrazolo[1,5-d][1,2,4]triazine
        Gene, Accession, CAS #CAS: 342652-67-9
        Catalog #3817/50
        Price
        Order / More InfoMRK 016 from TOCRIS BIOSCIENCE
        Product Specific ReferencesPubMed: 28275719
        產(chǎn)品資料
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