| 產(chǎn)品詳情 |
| Edit |   |
| Product Name | PF 04671536 hydrochloride |
| Description | Potent and selective PDE8B/8A inhibitor ( IC50 values are 1.3 and 1.9 nM, respectively). Exhibits selectivity for PDE8A/B over other PDEs (IC50 values are >10 μM) and a range of other targets. Increases glucose-dependent insulin secretion from human pacreatic islet cells. Orally bioavailable. Purity 98%. MW (observed): 382.87 |
| Size | 25 mg |
| Concentration | n/a |
| Applications | n/a |
| Other Names | 5-Methyl-3-[[(2R)-4-(2-thiazolylmethyl)-2-morpholinyl]methyl]-3H-1,2,3-triazolo[4,5-d]pyrimidin-7-amine hydrochloride |
| Gene, Accession, CAS # | CAS: 1305116-67-9 |
| Catalog # | 6024/25 |
| Price | |
| Order / More Info | PF 04671536 hydrochloride from TOCRIS BIOSCIENCE
|
| Product Specific References | n/a |
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